CULLETTA, Giulia
CULLETTA, Giulia
Scienze e Tecnologie Biologiche Chimiche e Farmaceutiche
A definitive pharmacophore modelling study on CDK2 ATP pocket binders: Tracing the path of new virtual high-throughput screenings
2020-01-01 Tutone M.; Culletta G.; Livecchi L.; Almerico A.M.
Aminoquinolines: Fluorescent sensors to DNA – A minor groove probe. Experimental and in silico studies
2023-10-01 de Carvalho Bertozo L.; Tutone M.; Pastrello B.; da Silva-Filho L.C.; Culletta G.; Almerico A.M.; Farias Ximenes V.
CHA on CDK2: a way to identify the best pharmacophore model for the virtual screening of new inhibitors
Chaperoning system: Intriguing target to modulate the expression of CFTR in cystic fibrosis
2024-08-28 Scalia F.; Culletta G.; Barreca M.; Caruso Bavisotto C.; Bivacqua R.; D'Amico G.; Alberti G.; Spano' V.; Tutone M.; Almerico A.M.; Cappello F.; Montalbano A.; Barraja P.
Comparing molecular dynamics-derived pharmacophore models with docking: A study on CDK-2 inhibitors
2020-01-01 Culletta G.; Almerico A.M.; Tutone M.
Evaluation of the IKKβ Binding of Indicaxanthin by Induced-Fit Docking, Binding Pose Metadynamics, and Molecular Dynamics
2021-09-10 Allegra M.; Tutone M.; Tesoriere L.; Attanzio A.; Culletta G.; Almerico A.M.
Exploring the new non-covalent immunoproteasome inhibitors of β1i /β5i subunits: Virtual screening and in vitro test
2023-01-01 Giulia Culletta; Marco Tutone; Ugo Perricone; Carla Di Chio; Anna Maria Almerico; Maria Zappalà
Exploring the non-covalent ligand-binding mechanism on immunoproteasome by enhanced Molecular Dynamics
2021-01-01 Culletta Giulia; Zappalà Maria; Ettari Roberta; Almerico Anna Maria; Tutone Marco
Exploring the SARS-CoV-2 proteome in the search of potential inhibitors via structure-based pharmacophore modeling/docking approach
2020-01-01 Culletta G.; Gulotta M.R.; Perricone U.; Zappala M.; Almerico A.M.; Tutone M.
Fighting Antibiotic Resistance: New Pyrimidine-Clubbed Benzimidazole Derivatives as Potential DHFR Inhibitors
2023-01-04 Haque, M.; Marathakam, Akash; Rana, Ritesh; Almehmadi, Samar; Tambe, Vishal; Charde, Manoj; Islam, Fahadul; Siddiqui, Falak; Culletta, Giulia; Almerico, Anna; Tutone, Marco; Khan, Sharuk
Immunoproteasome and Non-Covalent Inhibition: Exploration by Advanced Molecular Dynamics and Docking Methods
2021-07-02 Culletta, Giulia; Zappalà, Maria; Ettari, Roberta; Almerico, Anna Maria; Tutone, Marco
In Silico Design, Synthesis and Biological Evaluation of Anticancer Arylsulfonamide Endowed with Anti-Telomerase Activity
2022-01-10 Culletta G.; Allegra M.; Almerico A.M.; Restivo I.; Tutone M.
Indicaxanthin, a multi-target natural compound from Opuntia ficus-indica fruit: From its poly-pharmacological effects to biochemical mechanisms and molecular modelling studies
2019-01-01 Allegra, Mario; Tutone, Marco; Tesoriere, Luisa; Almerico, Anna Maria; Culletta, Giulia; Livrea, Maria Antonia; Attanzio, Alessandro
Investigating the inhibition of FTSJ1 a tryptophan tRNA-specific 2’-O-methyltransferase by NV TRIDs, as a mechanism of readthrough in nonsense mutated CFTR
2023-06-01 Pietro Salvatore Carollo; Marco Tutone; Giulia Culletta; Ignazio Fiduccia; Federica Corrao; Ivana Pibiri; Maria Grazia Zizzo; Raffaella Melfi; Andrea Pace; Anna Maria Almerico; Laura Lentini
INVESTIGATING THE NR2F2 STRUCTURE FOR DRUG REPURPOSING
2024-09-01 Giulia Culletta, Marco Tutone, Anna Maria Almerico
Natural products as non-covalent and covalent modulators of the KEAP1/NRF2 pathway exerting antioxidant effects
2024-03-26 Culletta, Giulia; Buttari, Brigitta; Arese, Marzia; Brogi, Simone; Almerico, Anna Maria; Saso, Luciano; Tutone, Marco
NEW TRANSLATIONAL READTHROUGH INDUCING DRUGS RESCUING NONSENSE MUTATED TP53: STRATEGIES AGAINST CANCER
Non-covalent immunoproteasome inhibitors: virtual screening and in vitro test on β1i /β5i subunits
2023-01-01 Giulia Culletta; Marco Tutone; Roberta Ettari; Ugo Perricone; Carla Di Chio; Anna Maria Almerico; Maria Zappalà
Pharmacophore-Based Design of New Chemical Scaffolds as Translational Readthrough-Inducing Drugs (TRIDs)
2020-01-01 Tutone M.; Pibiri I.; Perriera R.; Campofelice A.; Culletta G.; Melfi R.; Pace A.; Almerico A.M.; Lentini L.
Potential translational readthough inducin drugs: an optimized design and synthesis of new chemical scaffolds
Davide Ricci; Giulia Culletta; Marco Tutone; Ignazio Fiduccia; Emanuele Vitale; Carla Rizzo; Pietro Salvatore Carollo; Raffaella Melfi; Maria Grazia Zizzo; Laura Lentini; Ivana Pibiri