PARRINO, Barbara
PARRINO, Barbara
Scienze e Tecnologie Biologiche Chimiche e Farmaceutiche
1,2,4-Amino-triazine derivatives as pyruvate dehydrogenase kinase inhibitors: Synthesis and pharmacological evaluation
2023-01-23 Pecoraro, Camilla; De Franco, Michele; Carbone, Daniela; Bassani, Davide; Pavan, Matteo; Cascioferro, Stella; Parrino, Barbara; Cirrincione, Girolamo; Dall'Acqua, Stefano; Moro, Stefano; Gandin, Valentina; Diana, Patrizia
1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A
2021-01-01 Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana
1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase
2021-02-04 Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana
1,3,4-Oxadiazole and 1,3,4-Thiadiazole Nortopsentin Derivatives against Pancreatic Ductal Adenocarcinoma: Synthesis, Cytotoxic Activity, and Inhibition of CDK1
2023-07-19 Carbone, Daniela; Pecoraro, Camilla; Panzeca, Giovanna; Xu, Geng; Roeten, Margot S F; Cascioferro, Stella; Giovannetti, Elisa; Diana, Patrizia; Parrino, Barbara
1,3,5-Triazines: A promising scaffold for anticancer drugs development
2017-01-01 Cascioferro, S.; Parrino, B.; Spano', V.; Carbone, A.; Montalbano, A.; Barraja, P.; Diana, P.; Cirrincione, G.
11H‑Pyrido[3′,2′:4,5]pyrrolo[3,2‑c]cinnoline and Pyrido[3′,2′:4,5]pyrrolo[1,2‑c][1,2,3]benzotriazine: Two New Ring Systems with Antitumor Activity
2014-01-01 Parrino, B; Carbone, A; Muscarella, M; Spanò, V; Montalbano, A; Barraja, P; Salvador, A; Vedaldi, D; Cirrincione, G; Diana, P
2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent staphylococcal biofilm inhibitors
2019-04-01 Cascioferro, Stella; Parrino, Barbara; Petri, Giovanna Li; Cusimano, Maria Grazia; Schillaci, Domenico; Di Sarno, Veronica; Musella, Simona; Giovannetti, Elisa; Cirrincione, Girolamo; Diana, Patrizia
2-substituted-[1,3]thiazolo[4,5-e]isoindoles as kinases inhibiting compounds
2013-01-01 Spanò, V; Diana, P; Montalbano, A; Carbone, A; Parrino, B; Cirrincione, G; Barraja, P
3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma
2020-01-01 Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P.
3-[2-(1H-Indol-3-yl)-1,3-thiazol-4-yl)-1H-4-azaindole a new series of kinase inhibitors
2012-01-01 B. Parrino
3-[4-(1H-indol-3-yl)-1,3-thiazol-2-yl]-1H-pyrrolo[2,3-b]pyridines, nortopsentin Analogues with antiproliferative activity
2015-04-03 Parrino, B.; Carbone, A.; Di Vita, G.; Ciancimino, C.; Attanzio, A.; Spanò, V.; Montalbano, A.; Barraja, P.; Tesoriere, L.; Livrea, M.; Diana, P.; Cirrincione, G.
7-Azaindole-fused heterocycles with antitumor activity
2011-01-01 Diana, P; Barraja, P; Carbone, A; Parrino, B; Vedaldi, D; Salvador, A; Dall'Acqua, F; Brun, P; Cirrincione G
[1,2]oxazole[5,4-e]isoindoles as promising drugs for anticancer chemotherapy
2015-01-01 Spanò, V; Parrino, B; Carbone, A; Montalbano, A; Diana, P; Lopergolo, A; Pennati, M; Zaffaroni, N; Cirrincione, G; Barraja, P
[1,2]Oxazolo[5,4-e]isoindoles as promising tubulin polymerization inhibitors
2016-01-01 Spanò, V.; Pennati, M.; Parrino, B.; Carbone, A.; Montalbano, A.; Lopergolo, A.; Zuco, V.; Cominetti, D.; Diana, P.; Cirrincione, G.; Zaffaroni, N.; Barraja, P.
A Combination of Polymethoxyflavones from Citrus sinensis and Prenylflavonoids from Humulus lupulus Counteracts IL-1β-Induced Differentiated Caco-2 Cells Dysfunction via a Modulation of NF-κB/Nrf2 Activation
2023-08-16 Restivo, Ignazio; Basilicata, Manuela Giovanna; Giardina, Ilenia Concetta; Massaro, Alessandro; Pepe, Giacomo; Salviati, Emanuela; Pecoraro, Camilla; Carbone, Daniela; Cascioferro, Stella; Parrino, Barbara; Diana, Patrizia; Ostacolo, Carmine; Campiglia, Pietro; Attanzio, Alessandro; D’Anneo, Antonella; Pojero, Fanny; Allegra, Mario; Tesoriere, Luisa
A computational study to explore the molecular mechanisms behind the antiproliferative activity of Nortopsentin derivatives
2018-01-01 M.R. Gulotta, J. Lombino, B. Parrino, S.M. Cascioferro, P. Diana, A. Padova, G. Cirrincione, U. Perricone
A Facile Synthesis of Deaza-Analogues of the Bisindole Marine Alkaloid Topsentin
2013-01-01 Carbone, A; Spanò, V; Parrino, B; Ciancimino, C; Attanasi, OA; Favi, G
A New Oxadiazole-Based Topsentin Derivative Modulates Cyclin-Dependent Kinase 1 Expression and Exerts Cytotoxic Effects on Pancreatic Cancer Cells
2022-01-01 Camilla Pecoraro; Barbara Parrino; Stella Cascioferro; Adrian Puerta; Amir Avan; Godefridus J. Peters; Patrizia Diana; Elisa Giovannetti; Daniela Carbone
A Synthetic Derivative of Antimicrobial Peptide Holothuroidin 2 from Mediterranean Sea Cucumber (Holothuria tubulosa) in the Control of Listeria monocytogenes
2019-03-08 Cusimano, Maria Grazia; Spinello, Angelo; Barone, Giampaolo; Schillaci, Domenico; Cascioferro, Stella; Magistrato, Alessandra; Parrino, Barbara; Arizza, Vincenzo; Vitale, Maria
An efficient synthesis of pyrrolo[3',2':4,5]thiopyrano[3,2-b]pyridin-2-one: a new ring system of pharmaceutical interest
2012-01-01 Barraja, P; Diana, P; Spano, V; Montalbano, A; Carbone, A; Parrino, B; Cirrincione G