GIOVANNETTI, ELISA
GIOVANNETTI, ELISA
1,3,4-Oxadiazole and 1,3,4-Thiadiazole Nortopsentin Derivatives against Pancreatic Ductal Adenocarcinoma: Synthesis, Cytotoxic Activity, and Inhibition of CDK1
2023-07-19 Carbone, Daniela; Pecoraro, Camilla; Panzeca, Giovanna; Xu, Geng; Roeten, Margot S F; Cascioferro, Stella; Giovannetti, Elisa; Diana, Patrizia; Parrino, Barbara
3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma
2020-01-01 Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P.
Exploring Splicing Modulation as an Innovative Approach to Combat Pancreatic Cancer: SF3B1 Emerges as a Prognostic Indicator and Therapeutic Target
2024-01-01 Sciarrillo, Rocco; Terrana, Francesca; Comandatore, Annalisa; Supadmanaba, I Gede Putu; Wang, Bing; Hassouni, Btissame El; Mantini, Giulia; Jansen, Gerrit; Avan, Amir; Carbone, Daniela; Diana, Patrizia; Peters, Godefridus J; Morelli, Luca; Cloos, Jacqueline; Assaraf, Yehuda G; Giovannetti, Elisa
Exploring the therapeutic potential of a novel series of imidazothiadiazoles targeting focal adhesion kinase (FAK) for pancreatic cancer treatment: synthesis, mechanistic insights and promising antitumor and safety profile
2024-08-02 Pecoraro, Camilla; Carbone, Daniela; Scianò, Fabio; Terrana, Francesca; Xu, Geng; Bergonzini, Cecilia; Roeten, Margot S. F.; Cascioferro, Stella; Cirrincione, Girolamo; Diana, Patrizia; Giovannetti, Elisa; Parrino, Barbara
Exploring the therapeutic potential of focal adhesion kinase inhibition in overcoming chemoresistance in pancreatic ductal adenocarcinoma
2024-03-01 Sciano F.; Terrana F.; Pecoraro C.; Parrino B.; Cascioferro S.; Diana P.; Giovannetti E.; Carbone D.
Harnessing the tumor microenvironment: targeted cancer therapies through modulation of epithelial-mesenchymal transition
2025-01-13 Glaviano, A.; Lau, H.S.; Carter, L.M.; Lee, E.H.C.; Lam, H.Y.; Okina, E.; Tan, D.J.J.; Tan, W.; Ang, H.L.; Carbone, D.; Yee, M.Y.; Shanmugam, M.K.; Huang, X.Z.; Sethi, G.; Tan, T.Z.; Lim, L.H.K.; Huang, R.Y.; Ungefroren, H.; Giovannetti, E.; Tang, D.G.; Bruno, T.C.; Luo, P.; Andersen, M.H.; Qian, B.; Ishihara, J.; Radisky, D.C.; Elias, S.; Yadav, S.; Kim, M.; Robert, C.; Diana, P.; Schalper, K.A.; Shi, T.; Merghoub, T.; Krebs, S.; Kusumbe, A.P.; Davids, M.S.; Brown, J.R.; Kumar, A.P.
Impact of phospho-Akt expression on the clinical outcome and activity of gemcitabine and Akt inhibitors in pancreatic ductal adenocarcinoma
2017-01-01 Massihnia D.; Funel N.; Leon L.; Castiglia M.; Perez A.; Barraco N.; Listi A.; Galvano A.; Passiglia F.; Guarini A.; Calo V.; Rizzo S.; Castellana L.; Giovannetti E.; Russo A.
New Marine-Inspired Oxadiazole Derivatives for Use Against Pancreatic Ductal Adenocarcinoma
2025-08-14 Pecoraro, C.; Carbone, D.; Al Ostoot, F.H.M.; Vahabi, M.; Lencioni, G.; Diana, P.; Giovannetti, E.; Parrino, B.
Nortopsentins as Leads from Marine Organisms for Anticancer and Anti-Inflammatory Agent Development
2023-01-01 Pecoraro, C.; Terrana, F.; Panzeca, G.; Parrino, B.; Cascioferro, S.; Diana, P.; Giovannetti, E.; Carbone, D.
Novel Pyrazolo [1,5‐a]−1,3,5‐Triazine Derivatives as CDK7 Inhibitors: Synthesis and Biological Insights in Pancreatic Ductal Adenocarcinoma Models
2025-08-25 Carbone, D.; Terrana, F.; Sciuto, L.; Pecoraro, C.; Xu, G.; Cascioferro, S.; Cirrincione, G.; Peters, G.J.; Giovannetti, E.; Parrino, B.; Diana, P.
Synthesis and biological evaluation of a new class of azole urea compounds as Akt inhibitors with promising anticancer activity in pancreatic cancer models
2024-12-01 Camilla Pecoraro, Fabio Scianò, Daniela Carbone, Xu Geng, Deng Juan, Stella Cascioferro, Elisa Giovannetti, Patrizia Diana, Barbara Parrino
| Data di pubblicazione | Titolo | Autori | Tipologia | Autore(i) | File |
|---|---|---|---|---|---|
| 19-lug-2023 | 1,3,4-Oxadiazole and 1,3,4-Thiadiazole Nortopsentin Derivatives against Pancreatic Ductal Adenocarcinoma: Synthesis, Cytotoxic Activity, and Inhibition of CDK1 | Carbone, DanielaPecoraro, CamillaPanzeca, GiovannaCascioferro, StellaGiovannetti, ElisaDiana, PatriziaParrino, Barbara + | 01 - Contributo in rivista::1.01 Articolo in rivista | Carbone, Daniela; Pecoraro, Camilla; Panzeca, Giovanna; Xu, Geng; Roeten, Margot S F; Cascioferro, Stella; Giovannetti, Elisa; Diana, Patrizia; Parrino, Barbara | |
| 1-gen-2020 | 3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma | Cascioferro S.Li Petri G.Parrino B.Carbone D.Arizza V.Cirrincione G.Giovannetti E.Diana P. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P. | |
| 1-gen-2024 | Exploring Splicing Modulation as an Innovative Approach to Combat Pancreatic Cancer: SF3B1 Emerges as a Prognostic Indicator and Therapeutic Target | Terrana, FrancescaCarbone, DanielaDiana, PatriziaPeters, Godefridus JGiovannetti, Elisa + | 01 - Contributo in rivista::1.01 Articolo in rivista | Sciarrillo, Rocco; Terrana, Francesca; Comandatore, Annalisa; Supadmanaba, I Gede Putu; Wang, Bing; Hassouni, Btissame El; Mantini, Giulia; Jansen, Gerrit; Avan, Amir; Carbone, Daniela; Diana, Patrizia; Peters, Godefridus J; Morelli, Luca; Cloos, Jacqueline; Assaraf, Yehuda G; Giovannetti, Elisa | |
| 2-ago-2024 | Exploring the therapeutic potential of a novel series of imidazothiadiazoles targeting focal adhesion kinase (FAK) for pancreatic cancer treatment: synthesis, mechanistic insights and promising antitumor and safety profile | Pecoraro, CamillaCarbone, DanielaTerrana, FrancescaCascioferro, StellaCirrincione, GirolamoDiana, PatriziaGiovannetti, ElisaParrino, Barbara + | 01 - Contributo in rivista::1.01 Articolo in rivista | Pecoraro, Camilla; Carbone, Daniela; Scianò, Fabio; Terrana, Francesca; Xu, Geng; Bergonzini, Cecilia; Roeten, Margot S. F.; Cascioferro, Stella; Cirrincione, Girolamo; Diana, Patrizia; Giovannetti, Elisa; Parrino, Barbara | |
| 1-mar-2024 | Exploring the therapeutic potential of focal adhesion kinase inhibition in overcoming chemoresistance in pancreatic ductal adenocarcinoma | Terrana F.Pecoraro C.Parrino B.Cascioferro S.Diana P.Giovannetti E.Carbone D. + | 01 - Contributo in rivista::1.09 Review essay (rassegna critica) | Sciano F.; Terrana F.; Pecoraro C.; Parrino B.; Cascioferro S.; Diana P.; Giovannetti E.; Carbone D. | |
| 13-gen-2025 | Harnessing the tumor microenvironment: targeted cancer therapies through modulation of epithelial-mesenchymal transition | Glaviano, AntoninoCarbone, DanielaGiovannetti, ElisaDiana, Patrizia + | 01 - Contributo in rivista::1.09 Review essay (rassegna critica) | Glaviano, A.; Lau, H.S.; Carter, L.M.; Lee, E.H.C.; Lam, H.Y.; Okina, E.; Tan, D.J.J.; Tan, W.; Ang, H.L.; Carbone, D.; Yee, M.Y.; Shanmugam, M.K.; Huang, X.Z.; Sethi, G.; Tan, T.Z.; Lim, L.H.K.; Huang, R.Y.; Ungefroren, H.; Giovannetti, E.; Tang, D.G.; Bruno, T.C.; Luo, P.; Andersen, M.H.; Qian, B.; Ishihara, J.; Radisky, D.C.; Elias, S.; Yadav, S.; Kim, M.; Robert, C.; Diana, P.; Schalper, K.A.; Shi, T.; Merghoub, T.; Krebs, S.; Kusumbe, A.P.; Davids, M.S.; Brown, J.R.; Kumar, A.P. | |
| 1-gen-2017 | Impact of phospho-Akt expression on the clinical outcome and activity of gemcitabine and Akt inhibitors in pancreatic ductal adenocarcinoma | Massihnia D.Perez A.Barraco N.Listi A.Galvano A.Passiglia F.Guarini A.Calo V.Castellana L.Giovannetti E.Russo A. + | 01 - Contributo in rivista::1.05 Abstract in atti di convegno pubblicato in rivista | Massihnia D.; Funel N.; Leon L.; Castiglia M.; Perez A.; Barraco N.; Listi A.; Galvano A.; Passiglia F.; Guarini A.; Calo V.; Rizzo S.; Castellana L.; Giovannetti E.; Russo A. | |
| 14-ago-2025 | New Marine-Inspired Oxadiazole Derivatives for Use Against Pancreatic Ductal Adenocarcinoma | Pecoraro, CamillaCarbone, DanielaAl Ostoot, Fares Hezam MohammedDiana, PatriziaGiovannetti, ElisaParrino, Barbara + | 01 - Contributo in rivista::1.01 Articolo in rivista | Pecoraro, C.; Carbone, D.; Al Ostoot, F.H.M.; Vahabi, M.; Lencioni, G.; Diana, P.; Giovannetti, E.; Parrino, B. | |
| 1-gen-2023 | Nortopsentins as Leads from Marine Organisms for Anticancer and Anti-Inflammatory Agent Development | Pecoraro, C.Terrana, F.Panzeca, G.Parrino, B.Cascioferro, S.Diana, P.Giovannetti, E.Carbone, D. | 01 - Contributo in rivista::1.09 Review essay (rassegna critica) | Pecoraro, C.; Terrana, F.; Panzeca, G.; Parrino, B.; Cascioferro, S.; Diana, P.; Giovannetti, E.; Carbone, D. | |
| 25-ago-2025 | Novel Pyrazolo [1,5‐a]−1,3,5‐Triazine Derivatives as CDK7 Inhibitors: Synthesis and Biological Insights in Pancreatic Ductal Adenocarcinoma Models | Carbone, DanielaTerrana, FrancescaPecoraro, CamillaCascioferro, StellaCirrincione, GirolamoPeters, Godefridus J.Giovannetti, ElisaParrino, BarbaraDiana, Patrizia + | 01 - Contributo in rivista::1.01 Articolo in rivista | Carbone, D.; Terrana, F.; Sciuto, L.; Pecoraro, C.; Xu, G.; Cascioferro, S.; Cirrincione, G.; Peters, G.J.; Giovannetti, E.; Parrino, B.; Diana, P. | |
| 1-dic-2024 | Synthesis and biological evaluation of a new class of azole urea compounds as Akt inhibitors with promising anticancer activity in pancreatic cancer models | Camilla PecoraroDaniela CarboneStella CascioferroElisa GiovannettiPatrizia DianaBarbara Parrino + | 01 - Contributo in rivista::1.01 Articolo in rivista | Camilla Pecoraro, Fabio Scianò, Daniela Carbone, Xu Geng, Deng Juan, Stella Cascioferro, Elisa Giovannetti, Patrizia Diana, Barbara Parrino |