ALAMIA, Federica
ALAMIA, Federica
Scienze e Tecnologie Biologiche Chimiche e Farmaceutiche
A Hybrid In Silico Approach for Identifying Dual VEGFR/RAS Inhibitors as Potential Anticancer and Anti-Angiogenic Agents
2025-10-18 Bono, A.; La Monica, G.; Alamia, F.; Tocco, D.; Lauria, A.; Martorana, A.
A novel in silico approach for identifying multi-target JAK/STAT inhibitors as anticancer agents
2024-11-23 Bono, Alessia; La Monica, Gabriele; Alamia, Federica; Lauria, Antonino; Martorana, Annamaria
Bioisosteric heterocyclic analogues of natural bioactive flavonoids by scaffold-hopping approaches: State-of-the-art and perspectives in medicinal chemistry
2024-07-15 La Monica, Gabriele; Bono, Alessia; Alamia, Federica; Lauria, Antonino; Martorana, Annamaria
Combinatorial chemistry-driven In silico design and computational evaluation of covalent peptidomimetic SARS-CoV-2 main protease inhibitors via structure-based virtual screening and multivariate analysis
2025-06-01 Bono, Alessia; La Monica, Gabriele; Alamia, Federica; Mingoia, Francesco; Martorana, Annamaria; Lauria, Antonino
COVALENT INHIBITION IN TRIPLE-NEGATIVE BREAST CANCER: DESIGN, SYNTHESIS AND BIOLOGICAL PROFILING OF ACRYLAMIDE-BASED QUINOLINES
2025-09-14 La Monica, G.; Occhipinti, C.; Alamia, F.; Bono, A.; Lauria, A.; Palumbo Piccionello, A.; D'Anneo, A.; Martorana, A.
Design and Synthesis of Novel Thieno[3,2-c]quinoline Compounds with Antiproliferative Activity on RET-Dependent Medullary Thyroid Cancer Cells
2023-09-26 La Monica, Gabriele; Pizzolanti, Giuseppe; Baiamonte, Concetta; Bono, Alessia; Alamia, Federica; Mingoia, Francesco; Lauria, Antonino; Martorana, Annamaria
Design, Synthesis, and In Silico Insights of new 4‐Piperazinylquinolines as Antiproliferative Agents against NCI Renal Cancer Cell Lines
2025-02-05 La Monica, Gabriele; Bono, Alessia; Alamia, Federica; Martorana, Annamaria; Lauria, Antonino
In Silico Design of Dual Estrogen Receptor and Hsp90 Inhibitors for ER-Positive Breast Cancer Through a Mixed Ligand/Structure-Based Approach
2024-12-21 La Monica, G.; Alamia, F.; Bono, A.; Mingoia, F.; Martorana, A.; Lauria, A.
In Silico Design of New Dual Inhibitors of SARS-CoV-2 MPRO through Ligand- and Structure-Based Methods
2023-05-06 Bono, Alessia; Lauria, Antonino; La Monica, Gabriele; Alamia, Federica; Mingoia, Francesco; Martorana, Annamaria
In silico lead optimization and synthesis of a new series of thieno[3,2-c]quinoline with antiproliferative activity on RET-dependent medullary thyroid cancer cells
2023-12-11 Gabriele La Monica; Giuseppe Pizzolanti; Concetta Baiamonte; Alessia Bono; Federica Alamia; Giuseppe Siragusa; Francesco Mingoia; Antonino Lauria; Annamaria Martorana
In Silico Mixed Ligand/Structure-Based Design of New CDK-1/PARP-1 Dual Inhibitors as Anti-Breast Cancer Agents
2023-09-06 Bono, Alessia; La Monica, Gabriele; Alamia, Federica; Mingoia, Francesco; Gentile, Carla; Peri, Daniele; Lauria, Antonino; Martorana, Annamaria
Innovative In Silico Method for Discovering Multi-Target JAK/STAT Inhibitors as Potential Anticancer Therapies
2024-12-02 Bono Alessia; La Monica Gabriele; Alamia Federica; Lauria Antonino; Martorana Annamaria
Machine learning model for predicting molecular activity using Molecular Descriptors and ElectroShape Descriptors - FL051
2024-11-14 Alessia Bono; Aras Asad; Marco Albanese; Richard Ian Cooper; Antonino Lauria; Gabriele La Monica; Federica Alamia; Annamaria Martorana; Paul William Finn
New small molecules for the Treatment of TNBC innovative Polypharmacological In Silico Approach
2024-06-04 Federica Alamia, Gabriele La Monica, Alessia Bono, Antonino Lauria, Annamaria Martorana.
Novel 6,7-dimethoxy-4-piperazinylquinoline derivatives as promising antibacterial agents against Staphylococcus aureus
2024-01-01 Federica Alamia, Gabriele La Monica, Alessia Bono, Antonino Lauria, Rosa Alduina, Annamaria Gallo, Annamaria MARTORANA
Novel Antibacterial 4-Piperazinylquinoline Hybrid Derivatives Against Staphylococcus aureus: Design, Synthesis, and In Vitro and In Silico Insights
2024-12-25 La Monica, Gabriele; Gallo, Annamaria; Bono, Alessia; Alamia, Federica; Lauria, Antonino; Alduina, Rosa; Martorana, Annamaria
Optimized imidazole-thieno[3,2-c]quinolines: promising antiproliferative compounds for thyroid and NCI60 cancer cells
2024-11-01 Gabriele La Monica, Alessia Bono, Federica Alamia, Antonino Lauria, Giuseppe Pizzolanti, Giuseppe Siragusa, Concetta Baiamonte, Annamaria Martorana
Scaffold-Hopping Strategies in Aurone Optimization: A Comprehensive Review of Synthetic Procedures and Biological Activities of Nitrogen and Sulfur Analogues
2024-06-13 La Monica, Gabriele; Alamia, Federica; Bono, Alessia; Lauria, Antonino; Martorana, Annamaria
Synthesis, in vitro exploration, and reactivity studies of 6-chloropyridin-2-yl benzoates as promising covalent fragments with antiviral and pro-apoptotic activities
2025-06-23 Bono, A.; La Monica, G.; Alamia, F.; Tocco, D.; Attanzio, A.; Restivo, I.; Pizzolanti, G.; Palumbo Piccionello, A.; Lauria, A.; Martorana, A.