| Nome |
# |
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N-(INDAZOLYL)BENZAMIDO DERIVATIVES AS CDK1 INHIBITORS: DESIGN, SYNTHESIS, BIOLOGICAL ACTIVITY, AND MOLECULAR DOCKING STUDIES, file e3ad891b-659b-da0e-e053-3705fe0a2b96
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274
|
|
Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[2E]-3-phenylprop-2-enoylamino}benzamides, file e3ad8919-0095-da0e-e053-3705fe0a2b96
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203
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Pirrolomicine che inibiscono la Sortasi A nelle infezioni sostenute da batteri Gram-positivi, file e3ad891c-8c9c-da0e-e053-3705fe0a2b96
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186
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Non-Classical Transformation of Benzendiazonium Hydrogen Sulfates. Access to 1,3-Dimethylisochromeno[4,3-c]pyrazol-5(1H)-one, a Potential Benzodiazepine Receptor Ligand, file e3ad8916-8d68-da0e-e053-3705fe0a2b96
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167
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Comparative studies of the Pschorr reaction in the pyrazole series. Access to the new dibenzo(e,g)pyrazolo(1,5-a)(1,3)diazocine system of pharmaceutical interest, file e3ad8918-0bcf-da0e-e053-3705fe0a2b96
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139
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Discovery of a new class of sortase a transpeptidase inhibitors to tackle gram-positive pathogens: 2-(2-phenylhydrazinylidene)alkanoic acids and related derivatives, file e3ad8919-1921-da0e-e053-3705fe0a2b96
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127
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5-Amino-1-phenyl-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid, file e3ad8915-a308-da0e-e053-3705fe0a2b96
|
125
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Progettazione e sintesi di nuovi derivati 4-chinazolinonici potenziali inibitori della diidrofolato reduttasi, file e3ad891c-b759-da0e-e053-3705fe0a2b96
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112
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Pharmaceutical potential of synthetic and natural pyrrolomycins, file e3ad8919-953a-da0e-e053-3705fe0a2b96
|
98
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|
Isoxazolo[3,4-d]pyridazin-7(6H)-one derivatives endowed with anti-proliferative Activity., file e3ad891a-6fe7-da0e-e053-3705fe0a2b96
|
88
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Synthesis and antirpoliferative activity of isoxazolo[3,4-d]pyridazin-7(6H)-one derivatives, file e3ad8916-eed9-da0e-e053-3705fe0a2b96
|
78
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Sintesi di un isostero del 3,5-dimetil-6-fenil-8-(trifluorometil)-5,6-diidropirazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one (CF3-TZP) con potenziale attività biologica, file e3ad891c-b5e6-da0e-e053-3705fe0a2b96
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53
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NUOVI DERIVATI 2-ACETAMMIDOBENZAMMIDICI:
ATTIVITÀ ANTIPROLIFERATIVA E POSSIBILE MECCANISMO DI AZIONE, file e3ad891b-7afa-da0e-e053-3705fe0a2b96
|
47
|
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Synthesized benzamido derivatives exert antiproliferative effects by DNA damage and ROS generation., file e3ad891a-2cee-da0e-e053-3705fe0a2b96
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43
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Sintesi e valutazione biologica di nuovi nitroderivati analoghi della pirrolomicina D attivi su Pseudomonas aeruginosa, file e3ad891c-6efb-da0e-e053-3705fe0a2b96
|
37
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4-(3H)-quinazolinones N-3 substituted with a five membered heterocycle: A promising scaffold towards bioactive molecules, file e3ad8926-be4b-da0e-e053-3705fe0a2b96
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28
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Synthesis and antiproliferative activities of two new analogs of tetrazepinones, file e3ad891a-cf58-da0e-e053-3705fe0a2b96
|
17
|
|
Synthesis and antiproliferative activity of 3-(2-cloroethyl)-5-methyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4-(3H)-one, file e3ad8927-ef4b-da0e-e053-3705fe0a2b96
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14
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ATTIVITÀ ANTIPROLIFERATIVA DI UN DERIVATO POLICICLICO CON STRUTTURA COMPLESSA, file e3ad8916-f4c2-da0e-e053-3705fe0a2b96
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13
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Synthesis of alkyl-5,8-dimethyl-6-phenyl-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-ones of pharmaceutical interest, file e3ad891e-22b0-da0e-e053-3705fe0a2b96
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11
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Chemical composition, cytotoxic effects, antimicrobial and antibiofilm activity of Artemisia arborescens (Vaill.) L. growing wild in the province of Agrigento, Sicily, Italy., file e3ad8928-3d9b-da0e-e053-3705fe0a2b96
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11
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Synthesis and antiproliferative activity of a natural like glucosyl polycyclic compound, file e3ad8916-e6f2-da0e-e053-3705fe0a2b96
|
9
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|
Synthesis and antiproliferative activity of 3-(2-cloroethyl)-5-methyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4-(3H)-one, file e3ad8917-d975-da0e-e053-3705fe0a2b96
|
9
|
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New complex polycyclic compounds: Synthesis, antiproliferative activity and mechanism of action, file e3ad8922-2f31-da0e-e053-3705fe0a2b96
|
9
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|
Synthesis, antiproliferative activity and possible mechanism of action of novel 2-acetamidobenzamides bearing the 2-phenoxy functionality, file e3ad891c-42f6-da0e-e053-3705fe0a2b96
|
8
|
|
Novel 4-(3-phenylpropionamido), 4-(2-phenoxyacetamido) and 4-(cinnamamido) substituted benzamides bearing the pyrazole or indazole nucleus: synthesis, biological evaluation and mechanism of action, file e3ad891e-4e0c-da0e-e053-3705fe0a2b96
|
8
|
|
Synthesis of alkyl-5,8-dimethyl-6-phenyl-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-ones of pharmaceutical interest, file e3ad8915-9bdb-da0e-e053-3705fe0a2b96
|
7
|
|
Recent advanced in bioactive systems containing pyrazole fused with a five membered heterocycle, file e3ad8917-e86b-da0e-e053-3705fe0a2b96
|
7
|
|
Sortase A Inhibitors: Recent Advances and Future Perspectives, file e3ad8919-8aaa-da0e-e053-3705fe0a2b96
|
7
|
|
A new class of phenylhydrazinylidene derivatives as inhibitors of Staphylococcus aureus biofilm formation, file e3ad8919-1924-da0e-e053-3705fe0a2b96
|
6
|
|
Synthesis and biofilm formation reduction of pyrazole-4-carboxamide derivatives in some Staphylococcus aureus strains, file e3ad8919-dda3-da0e-e053-3705fe0a2b96
|
6
|
|
Derivati policiclici con struttura complessa dotati di attività antiproliferativa, file e3ad891a-c79a-da0e-e053-3705fe0a2b96
|
6
|
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The Reactivity of 4’-Substituted Spiro[Isoindole-1,3’-pyrazoles] Derivatives: Substitution/Elimination Reactions and Access to Biaryl Derivatives, file e3ad891a-e1f7-da0e-e053-3705fe0a2b96
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6
|
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Synthesis and antiproliferative activity of a natural like glycoconjugate polycyclic compound, file e3ad8919-2d1c-da0e-e053-3705fe0a2b96
|
5
|
|
Recent discoveries of anticancer flavonoids, file e3ad891b-5b12-da0e-e053-3705fe0a2b96
|
4
|
|
The role of (E)-6-chloro-3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-styrylquinazolin-4(3H)-one in the modulation of cannabinoidergic system. A pilot study, file e3ad891d-a0db-da0e-e053-3705fe0a2b96
|
4
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Synthesis, benzodiazepine receptor binding and molecular modelling
of isochromeno[4,3-c]pyrazol-5(1H)-one derivatives, file e3ad8916-1a0c-da0e-e053-3705fe0a2b96
|
3
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Anthranilamide-based 2-phenylcyclopropane-1-carboxamides, 1,1'-biphenyl-4-carboxamides and 1,1'-biphenyl-2-carboxamides: Synthesis biological evaluation and mechanism of action, file e3ad891a-eae3-da0e-e053-3705fe0a2b96
|
3
|
|
Synthesis and antifungal activity of new N-(1-phenil-4-carbetoxypyrazol-5-yl)-N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides, file e3ad8915-f3fb-da0e-e053-3705fe0a2b96
|
2
|
|
Synthesis of substituted 3-amino-N-phenyl-1H-indazole-1-carboxamides endowed with antiproliferative activity, file e3ad8918-faf4-da0e-e053-3705fe0a2b96
|
2
|
|
Synthesis and biological activity of new anti-inflammatory compounds containing the 1,4-benzodioxine and/or pyrrole system, file e3ad891d-e832-da0e-e053-3705fe0a2b96
|
2
|
|
Comparative Structural Studies of 4-Diazopyrazole Derivatives by X-Ray Diffraction and Theoretical Investigation, file e3ad8915-9bda-da0e-e053-3705fe0a2b96
|
1
|
|
Synthesis and antioproliferative activity of new derivatives containing the policyclic sistem 5,7:7,13-dimethanopyrazolo[3,4-b]pyrazolo[3'.4':2,3]azepino[4,5-f]azocine, file e3ad8916-76d6-da0e-e053-3705fe0a2b96
|
1
|
|
Unexpected synthesis by a non-classical Pschorr reaction of 3,5-dimethyl-1-phenyl-1,5-dihydro-4H-pyrazolo[4,3-c]quinolin-4-one, with binding affinity for the central benzodiazepine receptor, file e3ad8916-9901-da0e-e053-3705fe0a2b96
|
1
|
|
Synthesis and antiproliferative activity of new derivatives containing the polycyclic system 5,7:7,13-dimethanopyrazolo[3,4-b]pyrazolo[3’,4’:2,3]azepino[4,5-f]azocine, file e3ad8916-9e68-da0e-e053-3705fe0a2b96
|
1
|
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Synthesis and antifungal activity of new N-isoxazolyl-2-iodobenzamides, file e3ad8918-0c93-da0e-e053-3705fe0a2b96
|
1
|
|
Synthesis and induction of G0-G1 phase arrest with apoptosis of 3,5-dimethyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one, file e3ad891c-8042-da0e-e053-3705fe0a2b96
|
1
|
|
Discovery of a new class of sortase a transpeptidase inhibitors to tackle gram-positive pathogens: 2-(2-phenylhydrazinylidene)alkanoic acids and related derivatives, file e3ad8922-231e-da0e-e053-3705fe0a2b96
|
1
|
|
4-(3H)-quinazolinones N-3 substituted with a five membered heterocycle: A promising scaffold towards bioactive molecules, file e3ad8926-a9c7-da0e-e053-3705fe0a2b96
|
1
|
| Totale |
1.992 |