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SYNTHESIS AND IN VITRO ANTILEUKEMIC ACTIVITY OF NEW 4-TRIAZENOPYRAZOLE DERIVATIVES
2004-01-01 DAIDONE G; MAGGIO B; RAFFA D; PLESCIA S; SCHILLACI D; RAIMONDI MV
SYNTHESIS, CYTOTOXICITY, AND INHIBITORY EFFECTS ON TUBULIN POLYMERIZATION OF A NEW 3-HETEROCYCLO SUBSTITUTED 2-STYRYLQUINAZOLINONES
2004-01-01 RAFFA D; EDLER MC; DAIDONE G; MAGGIO B; MERIKECH M; PLESCIA S; SCHILLACI D; BAI R; HAMEL E
SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF 7-SUBSTITUTED1-ETHYL-3,4,10-TRIMETHYL-1,10-DIHYDRO-11H-PYRAZOLO(3,4-c)(1,6)BENZODIAZOCIN-11-ONE: A NEW RING SYSTEM
2004-01-01 MIGLIARA O; PLESCIA S; DIANA P; DI STEFANO V; CAMARDA L; DALL'OLIO R
Nonclassical Pschorr and Sandmeyer Reactions in Pyrazole Series
2005-01-01 MAGGIO, B; DAIDONE, G; RAFFA, D; PLESCIA, S; BOMBIERI, G; MENEGHETTI, F
Unclassical Pschorr and Sandmeyer reactions in pyrazole series
2005-01-01 MAGGIO B; DAIDONE G; RAFFA D; PLESCIA S; BOMBIERI G; MENEGHETTI F
Synthesis of New Indazol-3-yl derivatives as CDK1 inhibitors
2006-01-01 RAFFA D; MAGGIO B; CASCIOFERRO S; PLESCIA S; RAIMONDI MV
CDK: LigandFit Enrichment Plot of Active Compounds in a Screening Dataset.
2006-01-01 RAFFA D; MAGGIO B; CASCIOFERRO S; PLESCIA S; RAIMONDI MV
Synthesis and biological activity of new anti-inflammatory compounds containing the 1,4-benzodioxine and/or pyrrole system
2007-01-01 HARRAK Y; ROSELL G; DAIDONE G; PLESCIA S; SCHILLACI D; PUJOL MD
Antileukemic activity of some new 3-amino-N-phenyl-(1H)-indazole-1-carboxamide derivatives
2007-01-01 RAFFA D; MAGGIO B; RAIMONDI MV; CASCIOFERRO S; GALLO G; DAIDONE G; PLESCIA S
Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamide derivatives
2007-01-01 RAFFA D; MAGGIO B; RAIMONDI MV; CASCIOFERRO S; GALLO G; DAIDONE G; PLESCIA S
Synthesis and anticancer activity of 3-amino-N-phenyl-1H-indazole-1-carboxamide and 1-(1H)indazol-3-yl-3-phenylureido derivatives
2007-01-01 RAFFA D; MAGGIO B; CASCIOFERRO S; RAIMONDI V; SCHILLACI D; GALLO G; DAIDONE G; PLESCIA S; MENEGHETTI F; BOMBIERI G; TOLOMEO M; DI CRISTINA A; GRIMAUDO S
Electronic ionization mass spectra of 3-(5'-(3'-methylisoxazol))- and 3-(3'-(5'-methylisoxazol)-2-styryl-4(3H)quinazolinones of pharmaceutical interest:an useful tool to distinguish the two isomeric series
2008-01-01 Casula,G;Ceraulo,L;Ferrugia,M;Filizzola,F;Plescia,S;Raffa,D
Comparative studies of the Pschorr reaction in the pyrazole series. Access to the new dibenzo(e,g)pyrazolo(1,5-a)(1,3)diazocine system of pharmaceutical interest
2008-01-01 MAGGIO, B; RAFFA, D; RAIMONDI, MV; CASCIOFERRO, S; PLESCIA, S; SABATINO, MA; BOMBIERI, G; MENEGHETTI, F; DAIDONE, G
SYNTHESIS AND BIOLOGICAL EVALUATION OF 2-PHENYL-3-[INDAZOL-3-YL]-4(3H)-QUINAZOLINONES
2008-01-01 CASULA, G; PLESCIA, S; RAFFA, D; PLESCIA, F; MAGGIO, B; DAIDONE, G; RAIMONDI, MV; BOMBIERI, G; CUSIMANO, MG
SYNTHETIC AND BIOLOGICAL EVALUATION OF SOME NEW 2-CINNAMAMIDOBENZAMIDES AS POTENTIAL ANTAGONIST OF THE HDM2-P53 PROTEIN-PROTEIN INTERACTIONS
2008-01-01 RAFFA D; PLESCIA S; CASCIOFERRO S; CUSIMANO MG; TOLOMEO M
Synthesis and biological evaluation of some new 2-cinnamidobenzamides as potential antagonist of the HDM2-p53 protein-protein interactions
2008-01-01 Raffa,D;Plescia,S;Cascioferro,S;Cusimano,MG;Tolomeo,M
Synthesis and COX inhibition of 7-R1-8-R2-1-ethyl-3,4-dimethyl-, 4,10-dihydro-1H-pyrazolo[3,4-c][1,5]benzodiazocine-5,11-diones
2009-01-01 Migliara, O; Raffa, D; Plescia, S; Cusimano, MG; Carbone, A
N-(INDAZOLYL)BENZAMIDO DERIVATIVES AS CDK1 INHIBITORS: DESIGN, SYNTHESIS, BIOLOGICAL ACTIVITY, AND MOLECULAR DOCKING STUDIES
2009-01-01 Raffa, D.; Maggio, B.; Cascioferro, S.; Raimondi, M.; Daidone, G.; Plescia, S.; Schillaci, D.; Cusimano, M.; TITONE LANZA DI SCALEA, L.; Colomba, C.; Tolomeo, M.
Pyrazolo[3,4-d]pyrimidine Derivatives as COX-2 Selective Inhibitors: Synthesis and Molecular Modelling Studies
2009-01-01 Raffa, D; Maggio, B; Plescia, F; Cascioferro, SM; Raimondi, MV; Plescia, S; Cusimano, MG
Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamides
2009-01-01 RAFFA, D; MAGGIO, B; CASCIOFERRO, SM; RAIMONDI, MV; SCHILLACI, D; GALLO, G; DAIDONE, G; PLESCIA, S; MENEGHETTI, F; BOMBIERI, G; DI CRISTINA, A; PIPITONE, RM; GRIMAUDO, S; TOLOMEO, M
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