Sfoglia per Autore
New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma
2020-01-01 GIOVANNA LI PETRI; CAMILLA PECORARO; ORNELLA RANDAZZO; SILVIA ZOPPI; STELLA MARIA CASCIOFERRO; BARBARA PARRINO; DANIELA CARBONE; BTISSAME EL HASSOUNI; ANDREA CAVAZZONI; NADIA ZAFFARONI; GIROLAMO CIRRINCIONE; PATRIZIA DIANA; GODEFRIDUS J. PETERS; ELISA GIOVANNETTI
Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation
2021-01-01 Anna Carbone; Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Domenico Schillaci; Maria Grazia Cusimano; Girolamo Cirrincione; Patrizia Diana
Therapeutic strategies to counteract antibiotic resistance in MRSA biofilm-associated infections
2021-01-01 Stella Cascioferro; Daniela Carbone; Barbara Parrino; Camilla Pecoraro; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana
CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin
2021-01-01 Di Franco, Simone; Parrino, Barbara; Gaggianesi, Miriam; Pantina, Vincenzo Davide; Bianca, Paola; Nicotra, Annalisa; Mangiapane, Laura Rosa; Lo Iacono, Melania; Ganduscio, Gloria; Veschi, Veronica; Brancato, Ornella Roberta; Glaviano, Antonino; Turdo, Alice; Pillitteri, Irene; Colarossi, Lorenzo; Cascioferro, Stella; Carbone, Daniela; Pecoraro, Camilla; Fiori, Micol Eleonora; De Maria, Ruggero; Todaro, Matilde; Screpanti, Isabella; Cirrincione, Girolamo; Diana, Patrizia; Stassi, Giorgio
1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A
2021-01-01 Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana
1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase
2021-02-04 Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana
Novel strategies in the war against antibiotic resistance
2021-03-01 Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Patrizia Diana
Nobiletin and Xanthohumol Sensitize Colorectal Cancer Stem Cells to Standard Chemotherapy
2021-08-04 Alice Turdo; Antonino Glaviano; Giacomo Pepe; Federica Calapà; Stefania Raimondo; Micol Eleonora Fiori; Daniela Carbone; Manuela Giovanna Basilicata: Veronica Di Sarno; Carmine Ostacolo; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Simone Di Franco; Diana Bellavia; Miriam Gaggianesi; Veronica Veschi; Melania Lo Iacono; Gloria Ganduscio; Vincenzo Davide Pantina; Laura Rosa Mangiapane; Maria Rita Bongiorno; Riccardo Alessandro; Matilde Todaro; Ruggero De Maria; Patrizia Diana; Pietro Campiglia; Giorgio Stassi
GSK3β as a novel promising target to overcome chemoresistance in pancreatic cancer
2021-08-12 Pecoraro C.; Faggion B.; Balboni B.; Carbone D.; Peters G.J.; Diana P.; Assaraf Y.G.; Giovannetti E.
Cyclin dependent kinase-1 (Cdk-1) inhibition as a novel therapeutic strategy against pancreatic ductal adenocarcinoma (pdac)
2021-08-30 Wijnen R.; Pecoraro C.; Carbone D.; Fiuji H.; Avan A.; Peters G.J.; Giovannetti E.; Diana P.
SF3B1 modulators affect key genes in metastasis and drug influx: a new approach to fight pancreatic cancer chemoresistance
2021-10-01 Ornella Randazzo; Stella M. Cascioferro; Camilla Pecoraro; Widad Ait Iddouch; Amir Avan; Barbara Parrino; Daniela Carbone; Ugo Perricone; Godefridus J. Peters; Patrizia Diana; Elisa Giovannetti
Hop-derived fraction rich in beta acids and prenylflavonoids regulates the inflammatory response in dendritic cells differently from quercetin: unveiling metabolic changes by mass spectrometry-based metabolomics
2021-12-21 Eduardo Sommella; Giulio Verna; Marina Liso; Emanuela Salviati; Tiziana Esposito; Daniela Carbone; Camilla Pecoraro; Marcello Chieppa; Pietro Campiglia
Eight-membered heterocycles with two heteroatoms in a 1,3-relationship of interest in medicinal chemistry
2022-01-01 Barbara Parrino; Stella Cascioferro; Daniela Carbone; Camilla Pecoraro; Girolamo Cirrincione; Patrizia Diana
Synthesis and cytotoxic activity of 3-[2-(1H-Indol-3-yl)-1,3-thiazol-4-yl]-1Hpyrrolo[3,2-c]pyridine hydrobromides, analogues of the marine alkaloid nortopsentin
2022-01-01 Camilla Pecoraro; Daniela Carbone; Daniele Aiello; Anna Carbone
A New Oxadiazole-Based Topsentin Derivative Modulates Cyclin-Dependent Kinase 1 Expression and Exerts Cytotoxic Effects on Pancreatic Cancer Cells
2022-01-01 Camilla Pecoraro; Barbara Parrino; Stella Cascioferro; Adrian Puerta; Amir Avan; Godefridus J. Peters; Patrizia Diana; Elisa Giovannetti; Daniela Carbone
SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL SMALL MOLECULES AS PROMISING ALTERNATIVE AGENTS TO COUNTERACT DRUG RESISTANCE IN CANCER AND MICROBIAL INFECTIONS
2022-03-15
Metabolomics-assisted discovery of a new anticancer GLS-1 inhibitor chemotype from a nortopsentin-inspired library: From phenotype screening to target identification
2022-04-15 Carbone D.; Vestuto V.; Ferraro M.R.; Ciaglia T.; Pecoraro C.; Sommella E.; Cascioferro S.; Salviati E.; Novi S.; Tecce M.F.; Amodio G.; Iraci N.; Cirrincione G.; Campiglia P.; Diana P.; Bertamino A.; Parrino B.; Ostacolo C.
Synthesis and Antioxidative Properties of 1,2,3,4-Tetrahydropyridine Derivatives with Different Substituents in 4-Position
2022-11-01 Aiello, Daniele; Jonas, Hendrik; Carbone, Anna; Carbone, Daniela; Pecoraro, Camilla; Tesoriere, Luisa; Köhler, Jens; Wünsch, Bernhard; Diana, Patrizia
PI3K/AKT/mTOR signaling transduction pathway and targeted therapies in cancer
2023-01-01 Antonino Glaviano; Aaron S. C. Foo; Hiu Y. Lam; Kenneth C. H. Yap; William Jacot; Robert H. Jones; Huiyan Eng; Madhumathy G. Nair; Pooyan Makvandi; Birgit Geoerger; Matthew H. Kulke; Richard D. Baird; Jyothi S. Prabhu; Daniela Carbone; Camilla Pecoraro; Daniel B. L. Teh; Gautam Sethi; Vincenzo Cavalieri; Kevin H. Lin; Nathalie R. Javidi‑Sharifi; Eneda Toska; Matthew S. Davids; Jennifer R. Brown; Patrizia Diana; Justin Stebbing; David A. Fruman; Alan P. Kumar
Nortopsentins as Leads from Marine Organisms for Anticancer and Anti-Inflammatory Agent Development
2023-01-01 Pecoraro, C.; Terrana, F.; Panzeca, G.; Parrino, B.; Cascioferro, S.; Diana, P.; Giovannetti, E.; Carbone, D.
Data di pubblicazione | Titolo | Autori | Tipologia | Autore(i) | File |
---|---|---|---|---|---|
1-gen-2020 | New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma | GIOVANNA LI PETRICAMILLA PECORAROORNELLA RANDAZZOSTELLA MARIA CASCIOFERROBARBARA PARRINODANIELA CARBONEGIROLAMO CIRRINCIONEPATRIZIA DIANA + | 01 - Contributo in rivista::1.01 Articolo in rivista | GIOVANNA LI PETRI; CAMILLA PECORARO; ORNELLA RANDAZZO; SILVIA ZOPPI; STELLA MARIA CASCIOFERRO; BARBARA PARRINO; DANIELA CARBONE; BTISSAME EL HASSOUNI; ANDREA CAVAZZONI; NADIA ZAFFARONI; GIROLAMO CIRRINCIONE; PATRIZIA DIANA; GODEFRIDUS J. PETERS; ELISA GIOVANNETTI | |
1-gen-2021 | Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation | Anna CarboneStella CascioferroBarbara ParrinoDaniela CarboneCamilla PecoraroDomenico SchillaciMaria Grazia CusimanoGirolamo CirrincionePatrizia Diana | 01 - Contributo in rivista::1.01 Articolo in rivista | Anna Carbone; Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Domenico Schillaci; Maria Grazia Cusimano; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | Therapeutic strategies to counteract antibiotic resistance in MRSA biofilm-associated infections | Stella CascioferroDaniela CarboneBarbara ParrinoCamilla PecoraroGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Daniela Carbone; Barbara Parrino; Camilla Pecoraro; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin | Di Franco, SimoneParrino, BarbaraGaggianesi, MiriamPantina, Vincenzo DavideNicotra, AnnalisaMangiapane, Laura RosaLo Iacono, MelaniaGanduscio, GloriaVeschi, VeronicaGlaviano, AntoninoTurdo, AliceCascioferro, StellaCarbone, DanielaPecoraro, CamillaTodaro, MatildeCirrincione, GirolamoDiana, PatriziaStassi, Giorgio + | 01 - Contributo in rivista::1.01 Articolo in rivista | Di Franco, Simone; Parrino, Barbara; Gaggianesi, Miriam; Pantina, Vincenzo Davide; Bianca, Paola; Nicotra, Annalisa; Mangiapane, Laura Rosa; Lo Iacono, Melania; Ganduscio, Gloria; Veschi, Veronica; Brancato, Ornella Roberta; Glaviano, Antonino; Turdo, Alice; Pillitteri, Irene; Colarossi, Lorenzo; Cascioferro, Stella; Carbone, Daniela; Pecoraro, Camilla; Fiori, Micol Eleonora; De Maria, Ruggero; Todaro, Matilde; Screpanti, Isabella; Cirrincione, Girolamo; Diana, Patrizia; Stassi, Giorgio | |
1-gen-2021 | 1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A | Barbara ParrinoDaniela CarboneStella CascioferroCamilla PecoraroMaria Grazia CusimanoDomenico SchillaciGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana | |
4-feb-2021 | 1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase | Daniela CarboneBarbara ParrinoStella CascioferroCamilla PecoraroGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana | |
1-mar-2021 | Novel strategies in the war against antibiotic resistance | Stella CascioferroBarbara ParrinoDaniela CarboneCamilla PecoraroPatrizia Diana | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Patrizia Diana | |
4-ago-2021 | Nobiletin and Xanthohumol Sensitize Colorectal Cancer Stem Cells to Standard Chemotherapy | Alice TurdoAntonino GlavianoStefania RaimondoDaniela CarboneBarbara ParrinoStella CascioferroCamilla PecoraroSimone Di FrancoMiriam GaggianesiVeronica VeschiMelania Lo IaconoGloria GanduscioVincenzo Davide PantinaLaura Rosa MangiapaneMaria Rita BongiornoRiccardo AlessandroMatilde TodaroPatrizia DianaGiorgio Stassi + | 01 - Contributo in rivista::1.01 Articolo in rivista | Alice Turdo; Antonino Glaviano; Giacomo Pepe; Federica Calapà; Stefania Raimondo; Micol Eleonora Fiori; Daniela Carbone; Manuela Giovanna Basilicata: Veronica Di Sarno; Carmine Ostacolo; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Simone Di Franco; Diana Bellavia; Miriam Gaggianesi; Veronica Veschi; Melania Lo Iacono; Gloria Ganduscio; Vincenzo Davide Pantina; Laura Rosa Mangiapane; Maria Rita Bongiorno; Riccardo Alessandro; Matilde Todaro; Ruggero De Maria; Patrizia Diana; Pietro Campiglia; Giorgio Stassi | |
12-ago-2021 | GSK3β as a novel promising target to overcome chemoresistance in pancreatic cancer | Pecoraro C.Carbone D.Diana P. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Pecoraro C.; Faggion B.; Balboni B.; Carbone D.; Peters G.J.; Diana P.; Assaraf Y.G.; Giovannetti E. | |
30-ago-2021 | Cyclin dependent kinase-1 (Cdk-1) inhibition as a novel therapeutic strategy against pancreatic ductal adenocarcinoma (pdac) | Pecoraro C.Carbone D.Diana P. + | 01 - Contributo in rivista::1.09 Review essay (rassegna critica) | Wijnen R.; Pecoraro C.; Carbone D.; Fiuji H.; Avan A.; Peters G.J.; Giovannetti E.; Diana P. | |
1-ott-2021 | SF3B1 modulators affect key genes in metastasis and drug influx: a new approach to fight pancreatic cancer chemoresistance | Ornella RandazzoStella M. CascioferroCamilla PecoraroBarbara ParrinoDaniela CarbonePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Ornella Randazzo; Stella M. Cascioferro; Camilla Pecoraro; Widad Ait Iddouch; Amir Avan; Barbara Parrino; Daniela Carbone; Ugo Perricone; Godefridus J. Peters; Patrizia Diana; Elisa Giovannetti | |
21-dic-2021 | Hop-derived fraction rich in beta acids and prenylflavonoids regulates the inflammatory response in dendritic cells differently from quercetin: unveiling metabolic changes by mass spectrometry-based metabolomics | Daniela CarboneCamilla Pecoraro + | 01 - Contributo in rivista::1.01 Articolo in rivista | Eduardo Sommella; Giulio Verna; Marina Liso; Emanuela Salviati; Tiziana Esposito; Daniela Carbone; Camilla Pecoraro; Marcello Chieppa; Pietro Campiglia | |
1-gen-2022 | Eight-membered heterocycles with two heteroatoms in a 1,3-relationship of interest in medicinal chemistry | Barbara ParrinoStella CascioferroDaniela CarboneCamilla PecoraroPatrizia Diana + | 02 - Contributo in volume::2.01 Capitolo o Saggio | Barbara Parrino; Stella Cascioferro; Daniela Carbone; Camilla Pecoraro; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2022 | Synthesis and cytotoxic activity of 3-[2-(1H-Indol-3-yl)-1,3-thiazol-4-yl]-1Hpyrrolo[3,2-c]pyridine hydrobromides, analogues of the marine alkaloid nortopsentin | Camilla PecoraroDaniela CarboneDaniele AielloAnna Carbone | 01 - Contributo in rivista::1.01 Articolo in rivista | Camilla Pecoraro; Daniela Carbone; Daniele Aiello; Anna Carbone | |
1-gen-2022 | A New Oxadiazole-Based Topsentin Derivative Modulates Cyclin-Dependent Kinase 1 Expression and Exerts Cytotoxic Effects on Pancreatic Cancer Cells | Camilla PecoraroBarbara ParrinoStella CascioferroPatrizia DianaDaniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Camilla Pecoraro; Barbara Parrino; Stella Cascioferro; Adrian Puerta; Amir Avan; Godefridus J. Peters; Patrizia Diana; Elisa Giovannetti; Daniela Carbone | |
15-mar-2022 | SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL SMALL MOLECULES AS PROMISING ALTERNATIVE AGENTS TO COUNTERACT DRUG RESISTANCE IN CANCER AND MICROBIAL INFECTIONS | PECORARO, Camilla | 04 - Tesi di dottorato::4.2 Tesi di dottorato | - | |
15-apr-2022 | Metabolomics-assisted discovery of a new anticancer GLS-1 inhibitor chemotype from a nortopsentin-inspired library: From phenotype screening to target identification | Carbone D.Ferraro M. R.Pecoraro C.Cascioferro S.Cirrincione G.Diana P.Parrino B. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Carbone D.; Vestuto V.; Ferraro M.R.; Ciaglia T.; Pecoraro C.; Sommella E.; Cascioferro S.; Salviati E.; Novi S.; Tecce M.F.; Amodio G.; Iraci N.; Cirrincione G.; Campiglia P.; Diana P.; Bertamino A.; Parrino B.; Ostacolo C. | |
1-nov-2022 | Synthesis and Antioxidative Properties of 1,2,3,4-Tetrahydropyridine Derivatives with Different Substituents in 4-Position | Aiello, DanieleJonas, HendrikCarbone, AnnaCarbone, DanielaPecoraro, CamillaTesoriere, LuisaDiana, Patrizia + | 01 - Contributo in rivista::1.01 Articolo in rivista | Aiello, Daniele; Jonas, Hendrik; Carbone, Anna; Carbone, Daniela; Pecoraro, Camilla; Tesoriere, Luisa; Köhler, Jens; Wünsch, Bernhard; Diana, Patrizia | |
1-gen-2023 | PI3K/AKT/mTOR signaling transduction pathway and targeted therapies in cancer | Antonino GlavianoDaniela CarboneCamilla PecoraroVincenzo CavalieriPatrizia Diana + | 01 - Contributo in rivista::1.09 Review essay (rassegna critica) | Antonino Glaviano; Aaron S. C. Foo; Hiu Y. Lam; Kenneth C. H. Yap; William Jacot; Robert H. Jones; Huiyan Eng; Madhumathy G. Nair; Pooyan Makvandi; Birgit Geoerger; Matthew H. Kulke; Richard D. Baird; Jyothi S. Prabhu; Daniela Carbone; Camilla Pecoraro; Daniel B. L. Teh; Gautam Sethi; Vincenzo Cavalieri; Kevin H. Lin; Nathalie R. Javidi‑Sharifi; Eneda Toska; Matthew S. Davids; Jennifer R. Brown; Patrizia Diana; Justin Stebbing; David A. Fruman; Alan P. Kumar | |
1-gen-2023 | Nortopsentins as Leads from Marine Organisms for Anticancer and Anti-Inflammatory Agent Development | Pecoraro, C.Terrana, F.Panzeca, G.Parrino, B.Cascioferro, S.Diana, P.Giovannetti, E.Carbone, D. | 01 - Contributo in rivista::1.09 Review essay (rassegna critica) | Pecoraro, C.; Terrana, F.; Panzeca, G.; Parrino, B.; Cascioferro, S.; Diana, P.; Giovannetti, E.; Carbone, D. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile