Sfoglia per Autore
Resistance to epidermal growth factor receptor inhibition in non-small cell lung cancer
2018-01-01 Nele Van Der Steen, Elisa Giovannetti, Daniela Carbone, Alessandro Leonetti, Christian D. Rolfo, Godefridus J. Peters
Synthesis of novel 1,2,4-oxadiazole topsentin analogs with antitumor activity
2019-01-01 BARBARA PARRINO, DANIELA CARBONE, STELLA CASCIOFERRO, GODEFRIDUS J. PETERS, GIROLAMO CIRRINCIONE, ELISA GIOVANNETTI, PATRIZIA DIANA
Biological Evaluation of the Antiproliferative and Anti-migratory Activity of a Series of 3-(6-Phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)-1H-indole Derivatives against Pancreatic Cancer Cells*
2019-01-01 Li Petri G.; Cascioferro S.; El Hassouni B.; Carbone D.; Parrino B.; Cirrincione G.; Peters G.J.; Diana P.; Giovannetti E.
Biological evaluation of new 1,2,4-oxadiazole topsentin analogs as anticancer agents
2019-01-01 Barbara Parrino, Daniela Carbone, Stella Cascioferro, Btissame El Hassouni, Godefridus J. Peters, Girolamo Cirrincione, Elisa Giovannetti, Patrizia Diana
Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance
2020-01-01 Stella Cascioferro; Barbara Parrino; Daniela Carbone; Domenico Schillaci; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana
Eight-membered heterocycles with two heteroatoms in a 1,5-relationship of interest in medicinal chemistry
2020-01-01 Parrino B.; Cascioferro S.; Carbone D.; Cirrincione G.; Diana P.
Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives
2020-01-01 Parrino B.; Carbone D.; Cirrincione G.; Diana P.; Cascioferro S.
3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma
2020-01-01 Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P.
Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells
2020-01-01 Stella Cascioferro; Giovanna Li Petri ; Barbara Parrino; Daniela Carbone; Niccola Funel; Cecilia Bergonzini; Giulia Mantini; Henk Dekker; Daan Geerke; Godefridus J. Peters; Girolamo Cirrincione; Elisa Giovannetti; Patrizia Diana
Open Sesame? : Biomarker Status of the Human Equilibrative Nucleoside Transporter-1 and Molecular Mechanisms Influencing its Expression and Activity in the Uptake and Cytotoxicity of Gemcitabine in Pancreatic Cancer
2020-01-01 Ornella Randazzo; Filippo Papini; Giulia Mantini; Alessandro Gregori; Barbara Parrino; Daniel S. K. Liu; Stella Cascioferro; Daniela Carbone; Godefridus J. Peters; Adam E. Frampton; Ingrid Garajova; Elisa Giovannetti
New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma
2020-01-01 GIOVANNA LI PETRI; CAMILLA PECORARO; ORNELLA RANDAZZO; SILVIA ZOPPI; STELLA MARIA CASCIOFERRO; BARBARA PARRINO; DANIELA CARBONE; BTISSAME EL HASSOUNI; ANDREA CAVAZZONI; NADIA ZAFFARONI; GIROLAMO CIRRINCIONE; PATRIZIA DIANA; GODEFRIDUS J. PETERS; ELISA GIOVANNETTI
Dynamic-shared pharmacophore approach as tool to design new allosteric PRC2 inhibitors, targeting EED binding pocket
2021-01-01 Jessica Lombino; Maria Rita Gulotta; Giada De Simone; Nedra Mekni; Maria De Rosa; Daniela Carbone; Barbara Parrino; Stella Maria Cascioferro; Patrizia Diana; Alessandro Padova; Ugo Perricone
Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation
2021-01-01 Anna Carbone; Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Domenico Schillaci; Maria Grazia Cusimano; Girolamo Cirrincione; Patrizia Diana
Therapeutic strategies to counteract antibiotic resistance in MRSA biofilm-associated infections
2021-01-01 Stella Cascioferro; Daniela Carbone; Barbara Parrino; Camilla Pecoraro; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana
CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin
2021-01-01 Di Franco, Simone; Parrino, Barbara; Gaggianesi, Miriam; Pantina, Vincenzo Davide; Bianca, Paola; Nicotra, Annalisa; Mangiapane, Laura Rosa; Lo Iacono, Melania; Ganduscio, Gloria; Veschi, Veronica; Brancato, Ornella Roberta; Glaviano, Antonino; Turdo, Alice; Pillitteri, Irene; Colarossi, Lorenzo; Cascioferro, Stella; Carbone, Daniela; Pecoraro, Camilla; Fiori, Micol Eleonora; De Maria, Ruggero; Todaro, Matilde; Screpanti, Isabella; Cirrincione, Girolamo; Diana, Patrizia; Stassi, Giorgio
1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A
2021-01-01 Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana
Eight-membered heterocycles with two heteroatoms in a 1,2-relationship of interest in medicinal chemistry
2021-01-01 Barbara Parrino; Stella Cascioferro; Daniela Carbone; Girolamo Cirrincione; Patrizia Diana
Analysis of the metabolic switch induced by the spirulina peptide SP6 in high fat diet ApoE-/-mice model: A direct infusion FT-ICR-MS based approach
2021-01-01 Eduardo Sommella; Albino Carrizzo; Fabrizio Merciaia; Veronica Di Sarno; Daniela Carbone; Massimiliano De Lucia; Simona Musella; Carmine Vecchione; Pietro Campiglia
1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase
2021-02-04 Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana
Novel strategies in the war against antibiotic resistance
2021-03-01 Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Patrizia Diana
Data di pubblicazione | Titolo | Autori | Tipologia | Autore(i) | File |
---|---|---|---|---|---|
1-gen-2018 | Resistance to epidermal growth factor receptor inhibition in non-small cell lung cancer | Daniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Nele Van Der Steen, Elisa Giovannetti, Daniela Carbone, Alessandro Leonetti, Christian D. Rolfo, Godefridus J. Peters | |
1-gen-2019 | Synthesis of novel 1,2,4-oxadiazole topsentin analogs with antitumor activity | BARBARA PARRINODANIELA CARBONESTELLA CASCIOFERROGIROLAMO CIRRINCIONEPATRIZIA DIANA + | 02 - Contributo in volume::2.07 Contributo in atti di convegno pubblicato in volume | BARBARA PARRINO, DANIELA CARBONE, STELLA CASCIOFERRO, GODEFRIDUS J. PETERS, GIROLAMO CIRRINCIONE, ELISA GIOVANNETTI, PATRIZIA DIANA | |
1-gen-2019 | Biological Evaluation of the Antiproliferative and Anti-migratory Activity of a Series of 3-(6-Phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)-1H-indole Derivatives against Pancreatic Cancer Cells* | Li Petri G.Cascioferro S.Carbone D.Parrino B.Cirrincione G.Diana P. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Li Petri G.; Cascioferro S.; El Hassouni B.; Carbone D.; Parrino B.; Cirrincione G.; Peters G.J.; Diana P.; Giovannetti E. | |
1-gen-2019 | Biological evaluation of new 1,2,4-oxadiazole topsentin analogs as anticancer agents | Barbara ParrinoDaniela CarboneStella CascioferroGirolamo CirrincionePatrizia Diana + | 02 - Contributo in volume::2.08 Abstract in atti di convegno pubblicato in volume | Barbara Parrino, Daniela Carbone, Stella Cascioferro, Btissame El Hassouni, Godefridus J. Peters, Girolamo Cirrincione, Elisa Giovannetti, Patrizia Diana | |
1-gen-2020 | Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance | Stella CascioferroBarbara ParrinoDaniela CarboneDomenico SchillaciGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Barbara Parrino; Daniela Carbone; Domenico Schillaci; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2020 | Eight-membered heterocycles with two heteroatoms in a 1,5-relationship of interest in medicinal chemistry | Parrino B.Cascioferro S.Carbone D.Cirrincione G.Diana P. | 02 - Contributo in volume::2.01 Capitolo o Saggio | Parrino B.; Cascioferro S.; Carbone D.; Cirrincione G.; Diana P. | |
1-gen-2020 | Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives | Parrino B.Carbone D.Cirrincione G.Diana P.Cascioferro S. | 01 - Contributo in rivista::1.01 Articolo in rivista | Parrino B.; Carbone D.; Cirrincione G.; Diana P.; Cascioferro S. | |
1-gen-2020 | 3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma | Cascioferro S.Li Petri G.Parrino B.Carbone D.Arizza V.Cirrincione G.Giovannetti E.Diana P. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P. | |
1-gen-2020 | Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells | Stella CascioferroGiovanna Li PetriBarbara ParrinoDaniela CarboneGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Giovanna Li Petri ; Barbara Parrino; Daniela Carbone; Niccola Funel; Cecilia Bergonzini; Giulia Mantini; Henk Dekker; Daan Geerke; Godefridus J. Peters; Girolamo Cirrincione; Elisa Giovannetti; Patrizia Diana | |
1-gen-2020 | Open Sesame? : Biomarker Status of the Human Equilibrative Nucleoside Transporter-1 and Molecular Mechanisms Influencing its Expression and Activity in the Uptake and Cytotoxicity of Gemcitabine in Pancreatic Cancer | Ornella RandazzoBarbara ParrinoStella CascioferroDaniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Ornella Randazzo; Filippo Papini; Giulia Mantini; Alessandro Gregori; Barbara Parrino; Daniel S. K. Liu; Stella Cascioferro; Daniela Carbone; Godefridus J. Peters; Adam E. Frampton; Ingrid Garajova; Elisa Giovannetti | |
1-gen-2020 | New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma | GIOVANNA LI PETRICAMILLA PECORAROORNELLA RANDAZZOSTELLA MARIA CASCIOFERROBARBARA PARRINODANIELA CARBONEGIROLAMO CIRRINCIONEPATRIZIA DIANA + | 01 - Contributo in rivista::1.01 Articolo in rivista | GIOVANNA LI PETRI; CAMILLA PECORARO; ORNELLA RANDAZZO; SILVIA ZOPPI; STELLA MARIA CASCIOFERRO; BARBARA PARRINO; DANIELA CARBONE; BTISSAME EL HASSOUNI; ANDREA CAVAZZONI; NADIA ZAFFARONI; GIROLAMO CIRRINCIONE; PATRIZIA DIANA; GODEFRIDUS J. PETERS; ELISA GIOVANNETTI | |
1-gen-2021 | Dynamic-shared pharmacophore approach as tool to design new allosteric PRC2 inhibitors, targeting EED binding pocket | Jessica LombinoMaria Rita GulottaDaniela CarboneBarbara ParrinoStella Maria CascioferroPatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Jessica Lombino; Maria Rita Gulotta; Giada De Simone; Nedra Mekni; Maria De Rosa; Daniela Carbone; Barbara Parrino; Stella Maria Cascioferro; Patrizia Diana; Alessandro Padova; Ugo Perricone | |
1-gen-2021 | Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation | Anna CarboneStella CascioferroBarbara ParrinoDaniela CarboneCamilla PecoraroDomenico SchillaciMaria Grazia CusimanoGirolamo CirrincionePatrizia Diana | 01 - Contributo in rivista::1.01 Articolo in rivista | Anna Carbone; Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Domenico Schillaci; Maria Grazia Cusimano; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | Therapeutic strategies to counteract antibiotic resistance in MRSA biofilm-associated infections | Stella CascioferroDaniela CarboneBarbara ParrinoCamilla PecoraroGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Daniela Carbone; Barbara Parrino; Camilla Pecoraro; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin | Di Franco, SimoneParrino, BarbaraGaggianesi, MiriamPantina, Vincenzo DavideNicotra, AnnalisaMangiapane, Laura RosaLo Iacono, MelaniaGanduscio, GloriaVeschi, VeronicaGlaviano, AntoninoTurdo, AliceCascioferro, StellaCarbone, DanielaPecoraro, CamillaTodaro, MatildeCirrincione, GirolamoDiana, PatriziaStassi, Giorgio + | 01 - Contributo in rivista::1.01 Articolo in rivista | Di Franco, Simone; Parrino, Barbara; Gaggianesi, Miriam; Pantina, Vincenzo Davide; Bianca, Paola; Nicotra, Annalisa; Mangiapane, Laura Rosa; Lo Iacono, Melania; Ganduscio, Gloria; Veschi, Veronica; Brancato, Ornella Roberta; Glaviano, Antonino; Turdo, Alice; Pillitteri, Irene; Colarossi, Lorenzo; Cascioferro, Stella; Carbone, Daniela; Pecoraro, Camilla; Fiori, Micol Eleonora; De Maria, Ruggero; Todaro, Matilde; Screpanti, Isabella; Cirrincione, Girolamo; Diana, Patrizia; Stassi, Giorgio | |
1-gen-2021 | 1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A | Barbara ParrinoDaniela CarboneStella CascioferroCamilla PecoraroMaria Grazia CusimanoDomenico SchillaciGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana | |
1-gen-2021 | Eight-membered heterocycles with two heteroatoms in a 1,2-relationship of interest in medicinal chemistry | Barbara ParrinoStella CascioferroDaniela CarbonePatrizia Diana + | 02 - Contributo in volume::2.01 Capitolo o Saggio | Barbara Parrino; Stella Cascioferro; Daniela Carbone; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | Analysis of the metabolic switch induced by the spirulina peptide SP6 in high fat diet ApoE-/-mice model: A direct infusion FT-ICR-MS based approach | Daniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Eduardo Sommella; Albino Carrizzo; Fabrizio Merciaia; Veronica Di Sarno; Daniela Carbone; Massimiliano De Lucia; Simona Musella; Carmine Vecchione; Pietro Campiglia | |
4-feb-2021 | 1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase | Daniela CarboneBarbara ParrinoStella CascioferroCamilla PecoraroGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana | |
1-mar-2021 | Novel strategies in the war against antibiotic resistance | Stella CascioferroBarbara ParrinoDaniela CarboneCamilla PecoraroPatrizia Diana | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Patrizia Diana |
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