Sfoglia per Autore
Resistance to epidermal growth factor receptor inhibition in non-small cell lung cancer
2018-01-01 Nele Van Der Steen, Elisa Giovannetti, Daniela Carbone, Alessandro Leonetti, Christian D. Rolfo, Godefridus J. Peters
Synthesis of novel 1,2,4-oxadiazole topsentin analogs with antitumor activity
2019-01-01 BARBARA PARRINO, DANIELA CARBONE, STELLA CASCIOFERRO, GODEFRIDUS J. PETERS, GIROLAMO CIRRINCIONE, ELISA GIOVANNETTI, PATRIZIA DIANA
Biological Evaluation of the Antiproliferative and Anti-migratory Activity of a Series of 3-(6-Phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)-1H-indole Derivatives against Pancreatic Cancer Cells*
2019-01-01 Li Petri G.; Cascioferro S.; El Hassouni B.; Carbone D.; Parrino B.; Cirrincione G.; Peters G.J.; Diana P.; Giovannetti E.
Biological evaluation of new 1,2,4-oxadiazole topsentin analogs as anticancer agents
2019-01-01 Barbara Parrino, Daniela Carbone, Stella Cascioferro, Btissame El Hassouni, Godefridus J. Peters, Girolamo Cirrincione, Elisa Giovannetti, Patrizia Diana
Eight-membered heterocycles with two heteroatoms in a 1,5-relationship of interest in medicinal chemistry
2020-01-01 Parrino B.; Cascioferro S.; Carbone D.; Cirrincione G.; Diana P.
New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma
2020-01-01 GIOVANNA LI PETRI; CAMILLA PECORARO; ORNELLA RANDAZZO; SILVIA ZOPPI; STELLA MARIA CASCIOFERRO; BARBARA PARRINO; DANIELA CARBONE; BTISSAME EL HASSOUNI; ANDREA CAVAZZONI; NADIA ZAFFARONI; GIROLAMO CIRRINCIONE; PATRIZIA DIANA; GODEFRIDUS J. PETERS; ELISA GIOVANNETTI
Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells
2020-01-01 Stella Cascioferro; Giovanna Li Petri ; Barbara Parrino; Daniela Carbone; Niccola Funel; Cecilia Bergonzini; Giulia Mantini; Henk Dekker; Daan Geerke; Godefridus J. Peters; Girolamo Cirrincione; Elisa Giovannetti; Patrizia Diana
Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance
2020-01-01 Stella Cascioferro; Barbara Parrino; Daniela Carbone; Domenico Schillaci; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana
Open Sesame? : Biomarker Status of the Human Equilibrative Nucleoside Transporter-1 and Molecular Mechanisms Influencing its Expression and Activity in the Uptake and Cytotoxicity of Gemcitabine in Pancreatic Cancer
2020-01-01 Ornella Randazzo; Filippo Papini; Giulia Mantini; Alessandro Gregori; Barbara Parrino; Daniel S. K. Liu; Stella Cascioferro; Daniela Carbone; Godefridus J. Peters; Adam E. Frampton; Ingrid Garajova; Elisa Giovannetti
Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives
2020-01-01 Parrino B.; Carbone D.; Cirrincione G.; Diana P.; Cascioferro S.
3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma
2020-01-01 Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P.
Dynamic-shared pharmacophore approach as tool to design new allosteric PRC2 inhibitors, targeting EED binding pocket
2021-01-01 Jessica Lombino; Maria Rita Gulotta; Giada De Simone; Nedra Mekni; Maria De Rosa; Daniela Carbone; Barbara Parrino; Stella Maria Cascioferro; Patrizia Diana; Alessandro Padova; Ugo Perricone
CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin
2021-01-01 Di Franco, Simone; Parrino, Barbara; Gaggianesi, Miriam; Pantina, Vincenzo Davide; Bianca, Paola; Nicotra, Annalisa; Mangiapane, Laura Rosa; Lo Iacono, Melania; Ganduscio, Gloria; Veschi, Veronica; Brancato, Ornella Roberta; Glaviano, Antonino; Turdo, Alice; Pillitteri, Irene; Colarossi, Lorenzo; Cascioferro, Stella; Carbone, Daniela; Pecoraro, Camilla; Fiori, Micol Eleonora; De Maria, Ruggero; Todaro, Matilde; Screpanti, Isabella; Cirrincione, Girolamo; Diana, Patrizia; Stassi, Giorgio
1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A
2021-01-01 Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana
Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation
2021-01-01 Anna Carbone; Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Domenico Schillaci; Maria Grazia Cusimano; Girolamo Cirrincione; Patrizia Diana
Therapeutic strategies to counteract antibiotic resistance in MRSA biofilm-associated infections
2021-01-01 Stella Cascioferro; Daniela Carbone; Barbara Parrino; Camilla Pecoraro; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana
Eight-membered heterocycles with two heteroatoms in a 1,2-relationship of interest in medicinal chemistry
2021-01-01 Barbara Parrino; Stella Cascioferro; Daniela Carbone; Girolamo Cirrincione; Patrizia Diana
Analysis of the metabolic switch induced by the spirulina peptide SP6 in high fat diet ApoE-/-mice model: A direct infusion FT-ICR-MS based approach
2021-01-01 Eduardo Sommella; Albino Carrizzo; Fabrizio Merciaia; Veronica Di Sarno; Daniela Carbone; Massimiliano De Lucia; Simona Musella; Carmine Vecchione; Pietro Campiglia
1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase
2021-02-04 Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana
Novel strategies in the war against antibiotic resistance
2021-03-01 Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Patrizia Diana
Data di pubblicazione | Titolo | Autori | Tipologia | Autore(i) | File |
---|---|---|---|---|---|
1-gen-2018 | Resistance to epidermal growth factor receptor inhibition in non-small cell lung cancer | Daniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Nele Van Der Steen, Elisa Giovannetti, Daniela Carbone, Alessandro Leonetti, Christian D. Rolfo, Godefridus J. Peters | |
1-gen-2019 | Synthesis of novel 1,2,4-oxadiazole topsentin analogs with antitumor activity | BARBARA PARRINODANIELA CARBONESTELLA CASCIOFERROGIROLAMO CIRRINCIONEPATRIZIA DIANA + | 02 - Contributo in volume::2.07 Contributo in atti di convegno pubblicato in volume | BARBARA PARRINO, DANIELA CARBONE, STELLA CASCIOFERRO, GODEFRIDUS J. PETERS, GIROLAMO CIRRINCIONE, ELISA GIOVANNETTI, PATRIZIA DIANA | |
1-gen-2019 | Biological Evaluation of the Antiproliferative and Anti-migratory Activity of a Series of 3-(6-Phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)-1H-indole Derivatives against Pancreatic Cancer Cells* | Li Petri G.Cascioferro S.Carbone D.Parrino B.Cirrincione G.Diana P. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Li Petri G.; Cascioferro S.; El Hassouni B.; Carbone D.; Parrino B.; Cirrincione G.; Peters G.J.; Diana P.; Giovannetti E. | |
1-gen-2019 | Biological evaluation of new 1,2,4-oxadiazole topsentin analogs as anticancer agents | Barbara ParrinoDaniela CarboneStella CascioferroGirolamo CirrincionePatrizia Diana + | 02 - Contributo in volume::2.08 Abstract in atti di convegno pubblicato in volume | Barbara Parrino, Daniela Carbone, Stella Cascioferro, Btissame El Hassouni, Godefridus J. Peters, Girolamo Cirrincione, Elisa Giovannetti, Patrizia Diana | |
1-gen-2020 | Eight-membered heterocycles with two heteroatoms in a 1,5-relationship of interest in medicinal chemistry | Parrino B.Cascioferro S.Carbone D.Cirrincione G.Diana P. | 02 - Contributo in volume::2.01 Capitolo o Saggio | Parrino B.; Cascioferro S.; Carbone D.; Cirrincione G.; Diana P. | |
1-gen-2020 | New Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives Inhibit FAK Phosphorylation and Potentiate the Antiproliferative Effects of Gemcitabine Through Modulation of the Human Equilibrative Nucleoside Transporter-1 in Peritoneal Mesothelioma | GIOVANNA LI PETRICAMILLA PECORAROORNELLA RANDAZZOSTELLA MARIA CASCIOFERROBARBARA PARRINODANIELA CARBONEGIROLAMO CIRRINCIONEPATRIZIA DIANA + | 01 - Contributo in rivista::1.01 Articolo in rivista | GIOVANNA LI PETRI; CAMILLA PECORARO; ORNELLA RANDAZZO; SILVIA ZOPPI; STELLA MARIA CASCIOFERRO; BARBARA PARRINO; DANIELA CARBONE; BTISSAME EL HASSOUNI; ANDREA CAVAZZONI; NADIA ZAFFARONI; GIROLAMO CIRRINCIONE; PATRIZIA DIANA; GODEFRIDUS J. PETERS; ELISA GIOVANNETTI | |
1-gen-2020 | Imidazo[2,1-b] [1,3,4]thiadiazoles with antiproliferative activity against primary and gemcitabine-resistant pancreatic cancer cells | Stella CascioferroGiovanna Li PetriBarbara ParrinoDaniela CarboneGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Giovanna Li Petri ; Barbara Parrino; Daniela Carbone; Niccola Funel; Cecilia Bergonzini; Giulia Mantini; Henk Dekker; Daan Geerke; Godefridus J. Peters; Girolamo Cirrincione; Elisa Giovannetti; Patrizia Diana | |
1-gen-2020 | Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance | Stella CascioferroBarbara ParrinoDaniela CarboneDomenico SchillaciGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Barbara Parrino; Daniela Carbone; Domenico Schillaci; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2020 | Open Sesame? : Biomarker Status of the Human Equilibrative Nucleoside Transporter-1 and Molecular Mechanisms Influencing its Expression and Activity in the Uptake and Cytotoxicity of Gemcitabine in Pancreatic Cancer | Ornella RandazzoBarbara ParrinoStella CascioferroDaniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Ornella Randazzo; Filippo Papini; Giulia Mantini; Alessandro Gregori; Barbara Parrino; Daniel S. K. Liu; Stella Cascioferro; Daniela Carbone; Godefridus J. Peters; Adam E. Frampton; Ingrid Garajova; Elisa Giovannetti | |
1-gen-2020 | Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives | Parrino B.Carbone D.Cirrincione G.Diana P.Cascioferro S. | 01 - Contributo in rivista::1.01 Articolo in rivista | Parrino B.; Carbone D.; Cirrincione G.; Diana P.; Cascioferro S. | |
1-gen-2020 | 3-(6-Phenylimidazo [2,1-b][1,3,4]thiadiazol-2-yl)-1HIndole derivatives as new anticancer agents in the treatment of pancreatic ductal adenocarcinoma | Cascioferro S.Li Petri G.Parrino B.Carbone D.Arizza V.Cirrincione G.Giovannetti E.Diana P. + | 01 - Contributo in rivista::1.01 Articolo in rivista | Cascioferro S.; Li Petri G. ; Parrino B.; El Hassouni B.; Carbone D.; Arizza V.; Perricone U.; Padova A.; Funel N.; Peters G.J.; Cirrincione G.; Giovannetti E.; Diana P. | |
1-gen-2021 | Dynamic-shared pharmacophore approach as tool to design new allosteric PRC2 inhibitors, targeting EED binding pocket | Jessica LombinoMaria Rita GulottaDaniela CarboneBarbara ParrinoStella Maria CascioferroPatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Jessica Lombino; Maria Rita Gulotta; Giada De Simone; Nedra Mekni; Maria De Rosa; Daniela Carbone; Barbara Parrino; Stella Maria Cascioferro; Patrizia Diana; Alessandro Padova; Ugo Perricone | |
1-gen-2021 | CHK1 inhibitor sensitizes resistant colorectal cancer stem cells to nortopsentin | Di Franco, SimoneParrino, BarbaraGaggianesi, MiriamPantina, Vincenzo DavideNicotra, AnnalisaMangiapane, Laura RosaLo Iacono, MelaniaGanduscio, GloriaVeschi, VeronicaGlaviano, AntoninoTurdo, AliceCascioferro, StellaCarbone, DanielaPecoraro, CamillaTodaro, MatildeCirrincione, GirolamoDiana, PatriziaStassi, Giorgio + | 01 - Contributo in rivista::1.01 Articolo in rivista | Di Franco, Simone; Parrino, Barbara; Gaggianesi, Miriam; Pantina, Vincenzo Davide; Bianca, Paola; Nicotra, Annalisa; Mangiapane, Laura Rosa; Lo Iacono, Melania; Ganduscio, Gloria; Veschi, Veronica; Brancato, Ornella Roberta; Glaviano, Antonino; Turdo, Alice; Pillitteri, Irene; Colarossi, Lorenzo; Cascioferro, Stella; Carbone, Daniela; Pecoraro, Camilla; Fiori, Micol Eleonora; De Maria, Ruggero; Todaro, Matilde; Screpanti, Isabella; Cirrincione, Girolamo; Diana, Patrizia; Stassi, Giorgio | |
1-gen-2021 | 1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A | Barbara ParrinoDaniela CarboneStella CascioferroCamilla PecoraroMaria Grazia CusimanoDomenico SchillaciGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Barbara Parrino, Daniela Carbone, Stella Cascioferro, Camilla Pecoraro, Elisa Giovannetti, Dongmei Deng, Veronica Di Sarno, Simona Musella, Giulia Auriemma, Maria Grazia Cusimano, Domenico Schillaci, Girolamo Cirrincione, Patrizia Diana | |
1-gen-2021 | Thiazole Analogues of the Marine Alkaloid Nortopsentin as Inhibitors of Bacterial Biofilm Formation | Anna CarboneStella CascioferroBarbara ParrinoDaniela CarboneCamilla PecoraroDomenico SchillaciMaria Grazia CusimanoGirolamo CirrincionePatrizia Diana | 01 - Contributo in rivista::1.01 Articolo in rivista | Anna Carbone; Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Domenico Schillaci; Maria Grazia Cusimano; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | Therapeutic strategies to counteract antibiotic resistance in MRSA biofilm-associated infections | Stella CascioferroDaniela CarboneBarbara ParrinoCamilla PecoraroGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Daniela Carbone; Barbara Parrino; Camilla Pecoraro; Elisa Giovannetti; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | Eight-membered heterocycles with two heteroatoms in a 1,2-relationship of interest in medicinal chemistry | Barbara ParrinoStella CascioferroDaniela CarbonePatrizia Diana + | 02 - Contributo in volume::2.01 Capitolo o Saggio | Barbara Parrino; Stella Cascioferro; Daniela Carbone; Girolamo Cirrincione; Patrizia Diana | |
1-gen-2021 | Analysis of the metabolic switch induced by the spirulina peptide SP6 in high fat diet ApoE-/-mice model: A direct infusion FT-ICR-MS based approach | Daniela Carbone + | 01 - Contributo in rivista::1.01 Articolo in rivista | Eduardo Sommella; Albino Carrizzo; Fabrizio Merciaia; Veronica Di Sarno; Daniela Carbone; Massimiliano De Lucia; Simona Musella; Carmine Vecchione; Pietro Campiglia | |
4-feb-2021 | 1,2,4-Oxadiazole Topsentin Analogs with Antiproliferative Activity against Pancreatic Cancer Cells, Targeting GSK3β Kinase | Daniela CarboneBarbara ParrinoStella CascioferroCamilla PecoraroGirolamo CirrincionePatrizia Diana + | 01 - Contributo in rivista::1.01 Articolo in rivista | Daniela Carbone; Barbara Parrino; Stella Cascioferro; Camilla Pecoraro; Elisa Giovannetti; Veronica Di Sarno; Simona Musella; Giulia Auriemma; Girolamo Cirrincione; Patrizia Diana | |
1-mar-2021 | Novel strategies in the war against antibiotic resistance | Stella CascioferroBarbara ParrinoDaniela CarboneCamilla PecoraroPatrizia Diana | 01 - Contributo in rivista::1.01 Articolo in rivista | Stella Cascioferro; Barbara Parrino; Daniela Carbone; Camilla Pecoraro; Patrizia Diana |
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